SCHEMBL8551172

SCHEMBL8551172

Nc1cc(Br)ccc1C(=O)OC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.52
SIGMAR1 Q99720 3/20 0.48
OPRK1 P41145 1/20 0.47
KMT2A Q03164 1/20 0.47
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CHRM2 P08172 3/20 0.46
CHRM3 P20309 3/20 0.46
DRD2 P14416 2/20 0.45
DRD4 P21917 2/20 0.45
DRD3 P35462 2/20 0.45
SCN1A P35498 1/20 0.45
SCN2A Q99250 1/20 0.45
SCN3A Q9NY46 1/20 0.45
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8554127 0.99 BCHE (0.51) BCHESIGMAR1OPRK1KMT2AMAPT
SCHEMBL8553603 0.89 BCHE (0.54) BCHESIGMAR1OPRK1KMT2ADRD2
SCHEMBL8552042 0.88 BCHE (0.53) BCHESIGMAR1OPRK1
Hydrochloric Acid SCHEMBL8553924 0.88 BCHE (0.53) BCHESIGMAR1OPRK1KMT2ADRD2
SCHEMBL8550210 0.88 SLC6A12 (0.54) BCHESIGMAR1OPRK1MAPTDRD2
SCHEMBL8551366 0.87 BCHE (0.52) BCHESIGMAR1OPRK1DRD2DRD4
SCHEMBL8553705 0.87 BCHE (0.52) BCHESIGMAR1KMT2AMAPTCHRM2
SCHEMBL8550767 0.87 BCHE (0.52) BCHEOPRK1DRD2DRD4DRD3
Hydrochloric Acid SCHEMBL8550148 0.87 SLC6A12 (0.53) BCHESIGMAR1OPRK1MAPTDRD2
Hydrochloric Acid SCHEMBL8554134 0.87 BCHE (0.52) BCHESIGMAR1OPRK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed