SCHEMBL8553603

SCHEMBL8553603

Nc1ccc(C(=O)OC2CCN(Cc3ccccc3)CC2)c(N)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.54
OPRK1 P41145 2/20 0.52
SIGMAR1 Q99720 2/20 0.50
ACHE P22303 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
ADRA2A P08913 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
DRD2 P14416 1/20 0.48
ADRA2B P18089 1/20 0.48
ADRA2C P18825 1/20 0.48
DRD4 P21917 1/20 0.48
SLC6A2 P23975 1/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
ADRA1A P35348 1/20 0.48
DRD3 P35462 1/20 0.48
HTR2B P41595 1/20 0.48
CHRNA4 P43681 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8553924 0.99 BCHE (0.53) BCHEOPRK1SIGMAR1ACHECYP1A2
SCHEMBL8550210 0.90 SLC6A12 (0.54) BCHEOPRK1SIGMAR1ACHECYP1A2
SCHEMBL8552042 0.90 BCHE (0.53) BCHEOPRK1SIGMAR1SLC6A12
SCHEMBL8551172 0.89 BCHE (0.52) BCHEOPRK1SIGMAR1DRD2DRD4
SCHEMBL8551366 0.89 BCHE (0.52) BCHEOPRK1SIGMAR1ACHECYP1A2
SCHEMBL8550767 0.89 BCHE (0.52) BCHEOPRK1ACHECYP1A2CYP3A4
Hydrochloric Acid SCHEMBL8554134 0.89 BCHE (0.52) BCHEOPRK1SIGMAR1SLC6A12MEN1
Hydrochloric Acid SCHEMBL8550148 0.89 SLC6A12 (0.53) BCHEOPRK1SIGMAR1ACHECYP1A2
SCHEMBL8551180 0.88 BCHE (0.58) BCHEOPRK1SIGMAR1SCN1ASCN2A
Hydrochloric Acid SCHEMBL8549503 0.88 BCHE (0.51) BCHEOPRK1ACHECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN claimed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP claimed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN claimed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US claimed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO claimed
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed