SCHEMBL8550347

SCHEMBL8550347

CCCOc1ccc2c(c1)c(-c1ccc(SC)cc1)c(OC(=O)O)n2Cc1ccc2nsnc2c1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 12/20 0.66
EDNRA P25101 9/20 0.59
PLA2G2A P14555 5/20 0.36
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549940 0.92 EDNRB (0.61) EDNRBEDNRAKDM4EGAAHSD17B10
SCHEMBL6661772 0.91 EDNRB (0.79) EDNRBEDNRAPLA2G2A
SCHEMBL8592785 0.91 EDNRB (0.69) EDNRBEDNRAPLA2G2AKDM4EGAA
SCHEMBL8550822 0.89 EDNRB (0.66) EDNRBEDNRAPLA2G2AKDM4EGAA
SCHEMBL8550345 0.89 EDNRB (0.83) EDNRBEDNRA
SCHEMBL8551602 0.88 EDNRB (0.69) EDNRBEDNRAPLA2G2AKDM4EHSD17B10
SCHEMBL8549097 0.86 EDNRB (0.67) EDNRBEDNRAPLA2G2A
SCHEMBL8553472 0.85 EDNRB (0.81) EDNRBEDNRA
SCHEMBL8548888 0.85 EDNRB (0.65) EDNRBEDNRAPLA2G2A
SCHEMBL8552415 0.85 EDNRB (0.65) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed