SCHEMBL8550755

SCHEMBL8550755

O=c1[nH]cnc2cc(-c3ncc[nH]3)ccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
PARP1 P09874 9/20 0.54
CHEK1 O14757 2/20 0.54
PIM1 P11309 2/20 0.54
RPS6KA3 P51812 1/20 0.54
KDM4A O75164 1/20 0.47
KDM4B O94953 1/20 0.47
KDM5C P41229 1/20 0.47
KDM4C Q9H3R0 1/20 0.47
KDM5B Q9UGL1 1/20 0.47
KDM3A Q9Y4C1 1/20 0.47
PDPK1 O15530 1/20 0.47
CA12 O43570 1/20 0.47
ALOX15 P16050 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CA9 Q16790 1/20 0.47
TNKS2 Q9H2K2 1/20 0.47
KDR P35968 3/20 0.46
EPHB4 P54760 3/20 0.46
TEK Q02763 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8782182 0.88 ACVR1 (0.57) PARP1CHEK1PIM1ACVR1AKT1
SCHEMBL12476626 0.78 PARP1 (0.62) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL6922381 0.76 PARP1 (0.63) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL4973091 0.76 PARP1 (0.56) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL13266881 0.74 PARP1 (0.55) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL643424 0.74 ALDH1A1 (1.00) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL29898482 0.74 ALDH1A1 (1.00) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL28223920 0.73 PARP1 (0.54) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL30101160 0.72 PARP1 (0.57) ALDH1A1PARP1CHEK1PIM1RPS6KA3
SCHEMBL14143352 0.72 PARP1 (0.62) ALDH1A1PARP1CHEK1PIM1RPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880517-A1 QUINAZOLINE COMPOUNDS ZENECA LIMITED (GB) 1998-12-02 EP disclosed
WO-1997030044-A1 QUINAZOLINE COMPOUNDS ZENECA LIMITED (GB) 1997-08-21 WO disclosed