SCHEMBL8550922

SCHEMBL8550922

OCc1cc2c(N3CCN(Cc4ccccc4)CC3)cccc2s1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.51
DRD3 P35462 4/20 0.51
DRD4 P21917 4/20 0.51
HTR6 P50406 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
ADRA1D P25100 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NCF1 P14598 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8546517 0.99 DRD2 (0.50) DRD2DRD3DRD4HTR6MEN1
SCHEMBL8544808 0.88 MEN1 (0.51) DRD2MEN1KMT2AADRA1DADRA1A
Hydrochloric Acid SCHEMBL6017322 0.87 CYP2C9 (0.50) DRD2MEN1KMT2AADRA1DADRA1A
SCHEMBL6017105 0.86 OPRM1 (0.50) DRD2MEN1KMT2A
Hydrochloric Acid SCHEMBL8546495 0.85 OPRM1 (0.49) DRD2MEN1KMT2A
Hydrochloric Acid SCHEMBL6017149 0.84 DRD4 (0.47) DRD2DRD3DRD4MEN1KMT2A
SCHEMBL9050996 0.81 HTR1A (0.44) DRD2DRD3DRD4ADRA1DADRA1A
SCHEMBL6017224 0.81 HTR1A (0.49) DRD2ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL6017117 0.81 DRD2 (0.47) DRD2DRD3ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL8550084 0.80 HTR1A (0.48) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660832-B1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMA INC (US) 1998-01-14 EP disclosed
US-5436246-A Compounds for treatment of anxiety, depression, migraine, stroke, angina and hypertension MERRELL DOW PHARMACEUTICALS INC. 1995-07-25 US disclosed
EP-0660832-A1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-07-05 EP disclosed
WO-1994006789-A1 SEROTONIN RECEPTOR AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-31 WO disclosed