SCHEMBL8551031

SCHEMBL8551031

COc1cc(-c2cc(C(=O)Cl)nc(C(=O)Cl)c2)ccc1OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.53
HPGD P15428 2/20 0.53
RAB9A P51151 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
TSHR P16473 3/20 0.50
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
HSD17B10 Q99714 2/20 0.50
ABCB1 P08183 1/20 0.50
USP2 O75604 1/20 0.50
LMNA P02545 1/20 0.50
ERN1 O75460 1/20 0.49
MCL1 Q07820 1/20 0.49
PDE4A P27815 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
CTSV O60911 2/20 0.48
CTSL P07711 2/20 0.48
APP P05067 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545841 0.90 MCL1 (0.56) NPC1HPGDRAB9ASMN1; SMN2TSHR
Hydrochloric Acid SCHEMBL8551040 0.89 MCL1 (0.55) NPC1HPGDRAB9ASMN1; SMN2TSHR
SCHEMBL8545077 0.79 TSHR (0.53) NPC1HPGDRAB9ASMN1; SMN2TSHR
SCHEMBL12303132 0.79 KDM4E (0.60) NPC1HPGDRAB9ASMN1; SMN2TSHR
SCHEMBL341137 0.78 NPC1 (0.73) NPC1HPGDRAB9ASMN1; SMN2KDM4E
SCHEMBL21003759 0.77 NPC1 (0.56) NPC1HPGDRAB9ASMN1; SMN2TSHR
SCHEMBL8545773 0.77 TSHR (0.53) NPC1HPGDRAB9ASMN1; SMN2TSHR
SCHEMBL8546271 0.76 MEN1 (0.48) NPC1HPGDRAB9ASMN1; SMN2TSHR
SCHEMBL14278335 0.75 MEN1 (0.57) HPGDKDM4EALDH1A1HSD17B10LMNA
SCHEMBL2392671 0.75 NPC1 (0.60) NPC1HPGDRAB9ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525825-B1 Substituted dicarboxy pyridine compounds EG & G WALLAC OY (FI) 1998-12-09 EP disclosed
EP-0195413-B1 Substituted pyridine derivatives BAXTER DIAGNOSTICS INC (US) 1993-11-18 EP disclosed
EP-0525825-A2 Substituted dicarboxy pyridine compounds Dade MicroScan Inc. (US) 1993-02-03 EP disclosed
US-4761481-A FLUORESCENT CHELATES, AMINE ACID COMPOUNDS BAXTER TRAVENOL LABORATORIES, INC. (US) 1988-08-02 US disclosed
EP-0195413-A2 Substituted pyridine derivatives Baxter Diagnostics Inc. (US) 1986-09-24 EP disclosed