SCHEMBL8551130

SCHEMBL8551130

COC(=O)c1c(I)cccc1C(=O)c1ccc(F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
CYP2C19 P33261 2/20 0.51
CYP2D6 P10635 1/20 0.51
TSHR P16473 1/20 0.51
RAB9A P51151 4/20 0.47
KMT2A Q03164 4/20 0.47
NPC1 O15118 3/20 0.47
MEN1 O00255 2/20 0.47
MAPT P10636 2/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.43
GAA P10253 2/20 0.43
ATM Q13315 1/20 0.42
KDM4E B2RXH2 4/20 0.41
LMNA P02545 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549362 0.87 TDP1 (0.50) RAB9AKMT2AMEN1MAPTGAA
SCHEMBL21253254 0.87 CYP1A2 (0.55) CYP1A2CYP2C19CYP2D6TSHRRAB9A
SCHEMBL8549312 0.87 TSHR (0.50) CYP1A2CYP2C19CYP2D6TSHRKMT2A
SCHEMBL8551927 0.83 CYP1A2 (0.48) CYP1A2CYP2C19CYP2D6TSHRRAB9A
SCHEMBL8551443 0.83 ALDH1A1 (0.49) CYP1A2CYP2C19CYP2D6TSHRRAB9A
SCHEMBL8553845 0.81 CYP1A2 (0.46) CYP1A2CYP2C19CYP2D6TSHRRAB9A
SCHEMBL30631292 0.80 CA1 (0.53) TSHRKMT2AMEN1MAPTMAPK1
SCHEMBL1097335 0.80 CA1 (0.53) TSHRKMT2AMEN1MAPTMAPK1
SCHEMBL8549684 0.79 ALDH1A1 (0.49) CYP1A2CYP2C19CYP2D6TSHRRAB9A
SCHEMBL8550492 0.79 CYP1A2 (0.44) CYP1A2CYP2C19CYP2D6TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed