SCHEMBL8551443

SCHEMBL8551443

COC(=O)c1c(N)cccc1C(=O)c1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
HSD17B10 Q99714 2/20 0.49
CFTR P13569 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
TSHR P16473 1/20 0.48
CYP2C19 P33261 1/20 0.48
MAPT P10636 5/20 0.47
RAB9A P51151 5/20 0.47
NPC1 O15118 4/20 0.47
KMT2A Q03164 4/20 0.47
MEN1 O00255 2/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
KDM4E B2RXH2 3/20 0.45
HPGD P15428 2/20 0.45
IKBKB O14920 1/20 0.44
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28229993 0.90 ALDH1A1 (0.53) ALDH1A1HSD17B10CFTRTSHRMAPT
SCHEMBL8547980 0.87 ALDH1A1 (0.50) ALDH1A1HSD17B10CFTRTSHRMAPT
SCHEMBL8547750 0.87 MAPT (0.59) ALDH1A1HSD17B10CFTRTSHRMAPT
SCHEMBL21253254 0.87 CYP1A2 (0.55) ALDH1A1CYP1A2CYP2D6TSHRCYP2C19
SCHEMBL8547708 0.86 ALDH1A1 (0.49) ALDH1A1HSD17B10CFTRMAPTRAB9A
SCHEMBL8551130 0.83 CYP1A2 (0.51) ALDH1A1CYP1A2CYP2D6TSHRCYP2C19
SCHEMBL8551927 0.83 CYP1A2 (0.48) ALDH1A1CYP1A2CYP2D6TSHRCYP2C19
SCHEMBL8553845 0.81 CYP1A2 (0.46) ALDH1A1CYP1A2CYP2D6TSHRCYP2C19
SCHEMBL60709 0.80 ALDH1A1 (0.69) ALDH1A1HSD17B10CFTRTSHRMAPT
SCHEMBL30342070 0.80 ALDH1A1 (0.69) ALDH1A1HSD17B10CFTRTSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed