SCHEMBL8551483

SCHEMBL8551483

CCCOc1ccc(-c2ccc(OCC(O)CCc3cccnc3)cc2)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRB3 P13945 1/20 0.41
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.40
PTAFR P25105 2/20 0.38
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
PPARG P37231 1/20 0.37
LMNA P02545 2/20 0.37
FFAR1 O14842 1/20 0.37
PPARD Q03181 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8483096 1.00 NAMPT (0.43) NAMPTMEN1KMT2ACYP3A4CYP2D6
SCHEMBL8552537 0.85 CYP11B1 (0.43) MEN1KMT2ACYP3A4CYP19A1PTAFR
SCHEMBL8477182 0.85 CYP11B1 (0.43) MEN1KMT2ACYP3A4CYP19A1PTAFR
SCHEMBL8552140 0.81 MEN1 (0.45) MEN1KMT2ACYP3A4CYP2D6CYP19A1
SCHEMBL8476865 0.81 MEN1 (0.45) MEN1KMT2ACYP3A4CYP2D6CYP19A1
SCHEMBL8117055 0.81 GRIN1 (0.43) MEN1KMT2ACYP3A4CYP2D6ADRB1
SCHEMBL8483060 0.81 MEN1 (0.42) MEN1KMT2ACYP3A4CYP2D6CYP19A1
SCHEMBL8118428 0.81 MEN1 (0.42) MEN1KMT2ACYP3A4CYP2D6CYP19A1
SCHEMBL8118260 0.81 MEN1 (0.42) MEN1KMT2ACYP3A4CYP2D6CYP19A1
SCHEMBL7766546 0.79 CYP3A4 (0.39) NAMPTMEN1KMT2ACYP3A4ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed