SCHEMBL8551491

SCHEMBL8551491

CCCCOc1c(Br)cc(C(=O)OC)c(C(=O)OC)c1Br

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 4/20 0.49
THRB P10828 4/20 0.49
SMN1; SMN2 Q16637 4/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ESR1 P03372 2/20 0.40
POLB P06746 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
RAB9A P51151 2/20 0.40
MAPT P10636 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
PLA2G2A P14555 2/20 0.38
NPC1 O15118 1/20 0.37
S1PR2 O95136 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548592 0.92 THRA (0.50) THRATHRBSMN1; SMN2ALDH1A1MEN1
SCHEMBL8548248 0.91 THRA (0.49) THRATHRBSMN1; SMN2ALDH1A1MEN1
SCHEMBL8548540 0.85 THRA (0.44) THRATHRBSMN1; SMN2ALDH1A1ESR1
SCHEMBL8550905 0.81 HSD17B10 (0.45) ALDH1A1POLBMAPTKDM4EHPGD
SCHEMBL8549251 0.80 THRA (0.55) THRATHRBSMN1; SMN2ALDH1A1MEN1
SCHEMBL13664126 0.79 THRA (0.43) THRATHRBSMN1; SMN2ALDH1A1MEN1
SCHEMBL13664228 0.78 THRA (0.42) THRATHRBSMN1; SMN2ESR1L3MBTL1
SCHEMBL12697311 0.74 CYP1A2 (0.51) SMN1; SMN2ALDH1A1ESR1L3MBTL1RAB9A
SCHEMBL12588846 0.73 SCN9A (0.41) THRATHRBSMN1; SMN2ALDH1A1MEN1
SCHEMBL13664194 0.72 KDM4E (0.42) THRATHRBSMN1; SMN2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed