SCHEMBL8548540

SCHEMBL8548540

CCCCOc1c(Br)cc(C(=O)c2ccccc2)c(C(=O)OC)c1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 4/20 0.44
THRB P10828 4/20 0.44
CCNB2 O95067 2/20 0.42
CCNE2 O96020 2/20 0.42
CDK1 P06493 2/20 0.42
CCNB1 P14635 2/20 0.42
CCNE1 P24864 2/20 0.42
CDK2 P24941 2/20 0.42
CCNB3 Q8WWL7 2/20 0.42
PLA2G2A P14555 1/20 0.40
NR1H4 Q96RI1 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPT P10636 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
LMNA P02545 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548592 0.86 THRA (0.50) THRATHRBPLA2G2ASMN1; SMN2MAPT
SCHEMBL8551491 0.85 THRA (0.49) THRATHRBPLA2G2ASMN1; SMN2MAPT
SCHEMBL8549089 0.85 CCNE2 (0.38) THRATHRBCCNB2CCNE2CDK1
SCHEMBL8546447 0.84 HPGD (0.46) SMN1; SMN2MAPTL3MBTL1CYP1A2CYP2C19
SCHEMBL8548248 0.82 THRA (0.49) THRATHRBSMN1; SMN2MAPTL3MBTL1
SCHEMBL12765211 0.75 CCNE2 (0.48) THRATHRBCCNB2CCNE2CDK1
SCHEMBL8549251 0.75 THRA (0.55) THRATHRBPLA2G2ASMN1; SMN2AKR1C2
SCHEMBL28809090 0.73 RAB9A (0.47) PLA2G2ASMN1; SMN2MAPTL3MBTL1CYP1A2
SCHEMBL16364900 0.73 THRB (0.54) THRATHRBMAPTL3MBTL1CYP1A2
SCHEMBL8378478 0.72 TSHR (0.51) SMN1; SMN2MAPTL3MBTL1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed