SCHEMBL8548592

SCHEMBL8548592

CCCCOc1c(Br)cc(C(=O)O)c(C(=O)OC)c1Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 4/20 0.50
THRB P10828 4/20 0.50
CNR2 P34972 1/20 0.40
HSD17B10 Q99714 2/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 2/20 0.39
POLB P06746 1/20 0.39
ESR1 P03372 2/20 0.39
TSHR P16473 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MCL1 Q07820 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
PLA2G2A P14555 1/20 0.37
S1PR3 Q99500 1/20 0.36
PTPN11 Q06124 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551491 0.92 THRA (0.49) THRATHRBSMN1; SMN2MEN1KMT2A
SCHEMBL8549251 0.89 THRA (0.55) THRATHRBCNR2HSD17B10SMN1; SMN2
SCHEMBL8548248 0.88 THRA (0.49) THRATHRBSMN1; SMN2MEN1KMT2A
SCHEMBL8548540 0.86 THRA (0.44) THRATHRBSMN1; SMN2ALDH1A1ESR1
SCHEMBL8549323 0.82 HSD17B10 (0.54) HSD17B10SMN1; SMN2ALDH1A1POLBTSHR
SCHEMBL27579122 0.77 THRA (0.47) THRATHRBCNR2HSD17B10ESR1
SCHEMBL13664228 0.76 THRA (0.42) THRATHRBSMN1; SMN2ESR1TSHR
SCHEMBL13664126 0.74 THRA (0.43) THRATHRBCNR2SMN1; SMN2MEN1
SCHEMBL11929251 0.73 THRA (0.49) THRATHRBCNR2HSD17B10TSHR
SCHEMBL10658494 0.73 PTPN11 (0.46) THRATHRBSMN1; SMN2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed