SCHEMBL8551547

SCHEMBL8551547

O=c1[nH]nc(-c2ccc(F)cc2)c2cccc(I)c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ATM Q13315 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GRM2 Q14416 1/20 0.41
PDGFRB P09619 1/20 0.40
SERPINE1 P05121 1/20 0.40
MAPT P10636 2/20 0.40
TNKS O95271 3/20 0.38
TNKS2 Q9H2K2 3/20 0.38
PARP2 Q9UGN5 2/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
PARP1 P09874 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549237 0.86 NPSR1 (0.62) ALDH1A1SMN1; SMN2ATMNPSR1MAPT
SCHEMBL8547192 0.85 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2ATMNPSR1MAPT
SCHEMBL8552572 0.82 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2ATMNPSR1GRM2
SCHEMBL8551845 0.80 ROCK2 (0.48) ALDH1A1SMN1; SMN2ATMNPSR1GRM2
SCHEMBL8551923 0.78 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2ATMNPSR1GRM2
SCHEMBL7884963 0.78 ATM (0.73) ALDH1A1SMN1; SMN2ATMNPSR1GRM2
SCHEMBL443588 0.77 PDPK1 (0.51) ALDH1A1SMN1; SMN2PDGFRBKDM4EGAA
SCHEMBL9226004 0.77 ATM (0.49) ALDH1A1SMN1; SMN2ATMNPSR1GRM2
SCHEMBL8549626 0.74 AR (0.42) ALDH1A1ATMNPSR1MAPTKDM4E
SCHEMBL8547763 0.72 ADORA2A (0.38) ALDH1A1SMN1; SMN2NPSR1MAPTMAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed