SCHEMBL8551845

SCHEMBL8551845

O=c1[nH]nc(-c2ccc(F)cc2)c2cccc(C(F)(F)F)c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.48
NAMPT P43490 2/20 0.48
ALDH1A1 P00352 3/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NPSR1 Q6W5P4 2/20 0.43
ATM Q13315 1/20 0.43
AR P10275 1/20 0.42
ENPP1 P22413 1/20 0.41
P2RX7 Q99572 2/20 0.41
PARP1 P09874 2/20 0.40
GRM2 Q14416 1/20 0.40
KDM4E B2RXH2 3/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
MAPT P10636 3/20 0.38
MAP2K4 P45985 1/20 0.38
TNKS O95271 3/20 0.37
TNKS2 Q9H2K2 3/20 0.37
PARP2 Q9UGN5 2/20 0.37
GAA P10253 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551923 0.89 ALDH1A1 (0.43) ROCK2NAMPTALDH1A1SMN1; SMN2NPSR1
SCHEMBL8551517 0.89 NPSR1 (0.57) ROCK2NAMPTALDH1A1SMN1; SMN2NPSR1
SCHEMBL8548542 0.88 ROCK2 (0.47) ROCK2NAMPTALDH1A1SMN1; SMN2NPSR1
SCHEMBL8551547 0.80 ALDH1A1 (0.48) ROCK2NAMPTALDH1A1SMN1; SMN2NPSR1
SCHEMBL8552572 0.80 ALDH1A1 (0.48) ROCK2NAMPTALDH1A1SMN1; SMN2NPSR1
SCHEMBL1407266 0.80 SMN1; SMN2 (0.50) ROCK2NAMPTALDH1A1SMN1; SMN2ENPP1
SCHEMBL3707918 0.78 ROCK2 (0.57) ROCK2NAMPTALDH1A1NPSR1ATM
SCHEMBL30602968 0.78 PIK3CA (0.46) ROCK2NAMPTNPSR1ATMPARP1
SCHEMBL26615156 0.78 PIK3CA (0.46) ROCK2NAMPTNPSR1ATMPARP1
SCHEMBL7884963 0.76 ATM (0.73) ROCK2NAMPTALDH1A1SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed