SCHEMBL855163

SCHEMBL855163

O=C1OC(=O)c2c(Cl)c(Cl)cc(F)c21

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
TSHR P16473 2/20 0.50
MEN1 O00255 1/20 0.32
HSP90AA1 P07900 1/20 0.32
KMT2A Q03164 1/20 0.32
AHR P35869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13991787 0.83 TSHR (0.39) ALDH1A1TSHR
SCHEMBL855290 0.80 TSHR (0.56) ALDH1A1TSHRMEN1HSP90AA1KMT2A
SCHEMBL18789227 0.77 ALDH1A1 (0.65) ALDH1A1TSHRAHR
SCHEMBL855012 0.72 ALDH1A1 (0.41) ALDH1A1TSHR
SCHEMBL855118 0.72 TSHR (0.65) ALDH1A1TSHR
SCHEMBL854561 0.72 ALDH1A1 (0.41) ALDH1A1TSHRMEN1HSP90AA1KMT2A
SCHEMBL855571 0.71 CA1 (0.33) ALDH1A1TSHR
SCHEMBL30523206 0.71 CA1 (0.33) ALDH1A1TSHR
SCHEMBL855516 0.69 EPAS1 (0.34) ALDH1A1
SCHEMBL853556 0.69 ALDH1A1 (0.48) ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2433933-B1 PRODUCTION METHOD OF TRI- OR TETRAHALOGEN-SUBSTITUTED PHTHALIDE SUMITOMO CHEMICAL CO (JP) 2019-05-08 EP disclosed
US-8604221-B2 Production method of halogen-substituted phthalide SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2013-12-10 US disclosed
US-20120142946-A1 PRODUCTION METHOD OF HALOGEN-SUBSTITUTED PHTHALIDE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-06-07 US disclosed
EP-2433933-A1 PRODUCTION METHOD OF HALOGEN-SUBSTITUTED PHTHALIDE Sumitomo Chemical Company, Limited (JP) 2012-03-28 EP disclosed