SCHEMBL8551720

SCHEMBL8551720

O=C(OC1CCN(Cc2ccccc2)CC1)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.60
PGR P06401 1/20 0.59
CHRM2 P08172 1/20 0.59
ABCB1 P08183 1/20 0.59
HTR1A P08908 1/20 0.59
ADRA2A P08913 1/20 0.59
ADORA3 P0DMS8 1/20 0.59
CHRM1 P11229 1/20 0.59
DRD1 P21728 1/20 0.59
TBXA2R P21731 1/20 0.59
SLC6A2 P23975 1/20 0.59
SLC6A4 P31645 1/20 0.59
ADRA1A P35348 1/20 0.59
OPRM1 P35372 1/20 0.59
DRD3 P35462 1/20 0.59
SLC6A3 Q01959 1/20 0.59
KCNH2 Q12809 1/20 0.59
CACNA1C Q13936 1/20 0.59
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8553181 0.99 SIGMAR1 (0.59) SIGMAR1PGRCHRM2ABCB1HTR1A
SCHEMBL8549295 0.94 MEN1 (0.64) SIGMAR1PGRCHRM2ABCB1HTR1A
Hydrochloric Acid SCHEMBL8686857 0.93 MEN1 (0.62) SIGMAR1PGRCHRM2ABCB1HTR1A
SCHEMBL8551099 0.88 MAPT (0.66) SIGMAR1CHRM2POLBMAPTCYP2C9
SCHEMBL8551863 0.88 MAPT (0.69) SIGMAR1CHRM2POLBMAPTCYP2C9
Hydrochloric Acid SCHEMBL8555329 0.87 MAPT (0.68) SIGMAR1CHRM2MEN1KMT2APOLB
Hydrochloric Acid SCHEMBL8550717 0.87 MAPT (0.65) SIGMAR1CHRM2POLBMAPTCYP2C9
SCHEMBL8553740 0.84 ALDH1A1 (0.60) SIGMAR1PGRCHRM2ABCB1HTR1A
SCHEMBL8550490 0.83 BCHE (0.65) CHRM2MEN1KMT2A
Hydrochloric Acid SCHEMBL8555461 0.83 ALDH1A1 (0.59) SIGMAR1PGRCHRM2ABCB1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed