SCHEMBL8552060

SCHEMBL8552060

COC(=O)COc1ccc(C(=O)Nc2cn(C3CCN(C(=O)OC(C)(C)C)CC3)cn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 6/20 0.47
CDK5R1 Q15078 6/20 0.47
GPR119 Q8TDV5 5/20 0.44
KDM4E B2RXH2 1/20 0.42
PKM P14618 1/20 0.42
KMT2A Q03164 1/20 0.42
MAPT P10636 2/20 0.42
CTSD P07339 1/20 0.41
CTSE P14091 1/20 0.41
BACE1 P56817 1/20 0.41
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
THRB P10828 1/20 0.41
HDAC1 Q13547 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8594911 0.84 NR3C1 (0.47) KMT2AMAPTCTSDCTSEBACE1
Hydrochloric Acid SCHEMBL8553008 0.83 CDK5 (0.49) CDK5CDK5R1MAPTALDH1A1
SCHEMBL8592851 0.77 CYP2C9 (0.45) GPR119KDM4EKMT2AMAPTALDH1A1
SCHEMBL25626286 0.72 GPR119 (0.47) GPR119KDM4EMAPTCTSDCTSE
SCHEMBL8550973 0.71 GPR119 (0.51) GPR119CTSDCTSEBACE1ALDH1A1
SCHEMBL8473888 0.71 GPR119 (0.68) GPR119ALDH1A1
SCHEMBL8473886 0.71 GPR119 (0.68) GPR119ALDH1A1
SCHEMBL947678 0.71 GPR119 (0.50) GPR119KDM4EMAPTCTSDCTSE
SCHEMBL7369010 0.70 MAPT (0.59) GPR119KMT2AMAPTALDH1A1
SCHEMBL27460187 0.70 GPR119 (0.49) GPR119KDM4EMAPTCTSDCTSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed