SCHEMBL8552266

SCHEMBL8552266

OC1CCN(Cc2ccccc2Br)CC1

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.63
TSHR P16473 2/20 0.63
ATM Q13315 1/20 0.63
RECQL P46063 1/20 0.63
L3MBTL1 Q9Y468 1/20 0.63
CYP2A13 Q16696 1/20 0.60
MAPT P10636 1/20 0.57
KDM4E B2RXH2 2/20 0.54
LMNA P02545 1/20 0.54
SLC18A3 Q16572 2/20 0.53
SIGMAR1 Q99720 1/20 0.50
FAAH O00519 1/20 0.50
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27883990 0.81 MPO (0.72) ALDH1A1TSHRMAPTKDM4ESIGMAR1
SCHEMBL8554449 0.80 ALDH1A1 (0.56) ALDH1A1TSHRATMRECQLL3MBTL1
SCHEMBL7447200 0.80 CYP2A13 (0.70) ALDH1A1TSHRATMRECQLL3MBTL1
SCHEMBL8551996 0.79 CXCR4 (0.69) ALDH1A1ATMCYP2A13MAPTKDM4E
SCHEMBL8551446 0.79 ALDH1A1 (0.64) ALDH1A1ATMCYP2A13MAPTKDM4E
SCHEMBL8550581 0.79 MAPT (0.57) ALDH1A1TSHRMAPTKDM4ELMNA
SCHEMBL28361515 0.79 ALDH1A1 (0.58) ALDH1A1TSHRATMRECQLL3MBTL1
SCHEMBL28542706 0.79 ALDH1A1 (0.58) ALDH1A1TSHRATMRECQLL3MBTL1
SCHEMBL18356563 0.78 ALDH1A1 (0.71) ALDH1A1TSHRATMRECQLL3MBTL1
SCHEMBL27776365 0.78 KDM4E (0.46) ALDH1A1TSHRATMRECQLL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed