SCHEMBL8554449

SCHEMBL8554449

O=C(Cl)C1CCN(Cc2ccccc2Br)CC1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
TSHR P16473 2/20 0.56
ATM Q13315 1/20 0.56
RECQL P46063 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
KDM4E B2RXH2 3/20 0.55
LMNA P02545 1/20 0.55
SIGMAR1 Q99720 1/20 0.54
CYP2A13 Q16696 1/20 0.53
FAAH O00519 2/20 0.51
HPGD P15428 1/20 0.51
PARP1 P09874 1/20 0.47
PARP2 Q9UGN5 1/20 0.47
MEN1 O00255 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3290324 0.80 MEN1 (0.68) TSHRSIGMAR1FAAHMEN1KMT2A
SCHEMBL8552266 0.80 ALDH1A1 (0.63) ALDH1A1TSHRATMRECQLL3MBTL1
Hydrochloric Acid SCHEMBL7828669 0.78 MEN1 (0.66) TSHRSIGMAR1FAAHMEN1KMT2A
SCHEMBL1474753 0.78 SIGMAR1 (0.70) TSHRATMSIGMAR1MEN1KMT2A
SCHEMBL14456744 0.77 KMT2A (0.56) ALDH1A1TSHRKDM4ELMNAMEN1
SCHEMBL28542706 0.76 ALDH1A1 (0.58) ALDH1A1TSHRATMRECQLL3MBTL1
SCHEMBL8228144 0.75 KMT2A (0.54) ALDH1A1TSHRATMKDM4ELMNA
SCHEMBL3747521 0.75 FAAH (0.68) ALDH1A1TSHRATMRECQLL3MBTL1
SCHEMBL5016390 0.75 MEN1 (0.65) ALDH1A1TSHRKDM4EFAAHHPGD
SCHEMBL8550475 0.74 ALDH1A1 (0.59) ALDH1A1TSHRATMRECQLL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed