SCHEMBL8552357

SCHEMBL8552357

C=CCOC(=O)c1ccc(CSC2CC(=O)N2)o1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.36
MAPT P10636 4/20 0.36
CYP3A4 P08684 1/20 0.36
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
LMNA P02545 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 2/20 0.33
POLB P06746 2/20 0.33
HSD17B10 Q99714 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300761 0.82 SNCA (0.42) ALDH1A1CYP3A4CA1CA2MEN1
SCHEMBL8552652 0.82 HTT (0.52) ALDH1A1MAPTLMNAMEN1KMT2A
Allyl Alcohol SCHEMBL8437400 0.80 SNCA (0.40) ALDH1A1CYP3A4CA1CA2MEN1
SCHEMBL8441196 0.78 NPSR1 (0.35) CYP3A4CA1CA2MEN1KMT2A
SCHEMBL11497029 0.72 ALDH1A1 (0.53) ALDH1A1MAPTCYP3A4LMNAMEN1
SCHEMBL17513682 0.72 CYP3A4 (0.58) ALDH1A1MAPTCYP3A4LMNAMEN1
SCHEMBL6215267 0.72 CYP3A4 (0.47) ALDH1A1MAPTCYP3A4LMNAGAA
SCHEMBL4677464 0.72 CYP3A4 (0.47) ALDH1A1MAPTCYP3A4LMNAGAA
SCHEMBL8102643 0.71 TSHR (0.37) ALDH1A1CYP3A4CA1CA2MEN1
SCHEMBL8104182 0.68 TSHR (0.44) ALDH1A1CYP3A4CA1CA2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840725-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1998-05-13 EP disclosed
WO-1997002242-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-01-23 WO disclosed