SCHEMBL8552558

SCHEMBL8552558

[CH2]CCOc1c(C)cc(C#N)cc1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN8A Q9UQD0 2/20 0.40
MRGPRX4 Q96LA9 2/20 0.33
MAPT P10636 2/20 0.33
GRM5 P41594 2/20 0.32
ABCC3 O15438 1/20 0.32
ESR1 P03372 1/20 0.32
CYP1A2 P05177 1/20 0.32
PGR P06401 1/20 0.32
CHRM2 P08172 1/20 0.32
ABCB1 P08183 1/20 0.32
CYP3A4 P08684 1/20 0.32
ADRA2A P08913 1/20 0.32
CYP2D6 P10635 1/20 0.32
CHRM1 P11229 1/20 0.32
CYP2C9 P11712 1/20 0.32
DRD1 P21728 1/20 0.32
PTGS1 P23219 1/20 0.32
SLC6A2 P23975 1/20 0.32
ADORA1 P30542 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554425 0.91 SCN8A (0.43) SCN8AMRGPRX4MAPTGRM5ABCC3
SCHEMBL28412531 0.81 HTR1A (0.41) SCN8AMRGPRX4MAPTTTRALB
SCHEMBL8137092 0.81 SCN8A (0.41) SCN8AMAPTCYP1A2CYP2D6KMT2A
SCHEMBL347967 0.79 KDM4E (0.46) SCN8AMAPTESR1CYP1A2CYP2D6
SCHEMBL13480569 0.79 GPR35 (0.41) SCN8AMAPTGRM5CYP1A2CYP3A4
SCHEMBL9523339 0.78 SCN8A (0.39) SCN8AMAPTCYP1A2CYP2D6KMT2A
SCHEMBL8876567 0.78 SCN8A (0.39) SCN8AMAPTCYP1A2CYP2D6KMT2A
SCHEMBL72030 0.78 KMT2A (0.46) MAPTKMT2ALMNAALDH1A1
SCHEMBL5314384 0.78 FFAR4 (0.36) EGLN2
SCHEMBL24942168 0.77 KDM4E (0.49) SCN8ACYP1A2CYP2D6CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846986-A Therapeutic phenoxyalkylazoles and phenoxyalkylazines SANOFI (FR) 1998-12-08 US disclosed
US-5763461-A ANTIPICORNAVIRAL AGENTS SANOFI (FR) 1998-06-09 US disclosed
US-5721261-A TREATING PICORNAVIRUS INFECTIONS SANOFI PHARMACEUTICALS, INC. (US) 1998-02-24 US disclosed