SCHEMBL8552595

SCHEMBL8552595

CCOC(=O)CCCc1ccc2[nH]c(COc3ccc(Cl)cc3)nc2c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.42
CNR1 P21554 1/20 0.41
MAPT P10636 4/20 0.40
CYSLTR2 Q9NS75 1/20 0.40
CYSLTR1 Q9Y271 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPY1R P25929 1/20 0.39
CHEK1 O14757 1/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
P2RY12 Q9H244 1/20 0.39
PTPN11 Q06124 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551098 0.89 RAB9A (0.45) RAB9ASMN1; SMN2TDP1NPC1POLB
SCHEMBL8554095 0.87 NPY1R (0.58) NPY1R
SCHEMBL8555194 0.86 SMN1; SMN2 (0.47) RAB9ASMN1; SMN2TDP1NPC1POLB
SCHEMBL8553989 0.86 RAB9A (0.47) RAB9ASMN1; SMN2TDP1NPC1POLB
SCHEMBL8554128 0.85 RAB9A (0.46) RAB9ASMN1; SMN2TDP1NPC1POLB
SCHEMBL8553401 0.85 RAB9A (0.41) RAB9ASMN1; SMN2TDP1NPC1POLB
SCHEMBL8554479 0.82 NPY1R (0.45) MAPTNPY1RPRMT5DGAT2ALDH1A1
SCHEMBL8557031 0.81 RAB9A (0.46) RAB9ASMN1; SMN2TDP1NPC1POLB
SCHEMBL8550273 0.80 RAB9A (0.42) RAB9ASMN1; SMN2TDP1NPC1POLB
SCHEMBL8552889 0.80 RAB9A (0.42) RAB9ASMN1; SMN2TDP1NPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0871442-A1 BENZIMIDZOLYL NEUROPEPTIDE Y RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1998-10-21 EP disclosed
WO-1997025041-A1 BENZIMIDZOLYL NEUROPEPTIDE Y RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed