SCHEMBL8552602

SCHEMBL8552602

CC(C)(C)OC(=O)N1C(=O)CC(C(F)(F)F)C1CC1OCCO1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
GLA P06280 1/20 0.34
KLK7 P49862 5/20 0.33
USP2 O75604 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NR1H2 P55055 1/20 0.32
DPP4 P27487 1/20 0.31
NAMPT P43490 1/20 0.31
KLK5 Q9Y337 4/20 0.30
ATM Q13315 2/20 0.30
PRSS1 P07477 2/20 0.30
PRSS2 P07478 2/20 0.30
PRSS3 P35030 2/20 0.30
CETP P11597 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549243 0.79 KDM4E (0.32) KDM4EMAPTTHRBCHRM2CHRM1
SCHEMBL8551638 0.72 KLK7 (0.40) THRBKLK7SMN1; SMN2KLK5PRSS1
SCHEMBL22728246 0.70 NR1H2 (0.42) KDM4EMAPTTHRBCHRM2CHRM1
SCHEMBL16690469 0.69 NR1H2 (0.46) KDM4EMAPTTHRBCHRM2CHRM1
SCHEMBL3730644 0.68 NR1H2 (0.45) KDM4EMAPTTHRBCHRM2CHRM1
SCHEMBL16689228 0.68 CHRM2 (0.41) KDM4EMAPTTHRBCHRM2CHRM1
SCHEMBL8021097 0.68 CHRM2 (0.42) MAPTCHRM2CHRM1CHRM3GLA
SCHEMBL14140977 0.68 CHRM2 (0.40) KDM4EMAPTTHRBCHRM2CHRM1
SCHEMBL352414 0.68 CHRM2 (0.34) KDM4EMAPTTHRBCHRM2CHRM1
SCHEMBL22096750 0.67 CHRM2 (0.46) KDM4EMAPTTHRBCHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824523-A1 NITRIC OXIDE SYNTHASE INHIBITORS DERIVED FROM CYCLIC AMIDINES G.D. Searle & Co. (US) 1998-02-25 EP disclosed
WO-1996035677-A1 NITRIC OXIDE SYNTHASE INHIBITORS DERIVED FROM CYCLIC AMIDINES G.D. SEARLE & CO. (US) 1996-11-14 WO disclosed