SCHEMBL8552712

SCHEMBL8552712

Clc1nnc(-c2ccsc2)c2cccc(Br)c12

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ENPP1 P22413 1/20 0.38
TDO2 P48775 1/20 0.35
NQO2 P16083 1/20 0.33
CYP2A6 P11509 4/20 0.33
CYP2B6 P20813 2/20 0.33
CYP2E1 P05181 1/20 0.33
GAA P10253 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PDGFRB P09619 1/20 0.31
PDGFRA P16234 1/20 0.31
PDPK1 O15530 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549262 0.80 ALDH1A1 (0.41) CYP3A4CYP2C9CYP2C19PDPK1ADORA2A
SCHEMBL8551565 0.79 KMT2A (0.42) GAACYP3A4CYP2C9CYP2C19ADORA2A
SCHEMBL9253635 0.79 CYP2A6 (0.42) TDO2NQO2CYP2A6CYP2B6CYP2E1
SCHEMBL8371541 0.77 PLAU (0.42) ENPP1TDO2NQO2
SCHEMBL8551877 0.77 ESR1 (0.37) CYP3A4CYP2C9CYP2C19ADORA2AADORA1
Hydrochloric Acid SCHEMBL8553292 0.76 PLAU (0.41) TDO2NQO2
SCHEMBL8371540 0.75 CCNE2 (0.32) ENPP1TDO2NQO2
Hydrochloric Acid SCHEMBL8553284 0.74 CCNE2 (0.32) ENPP1
SCHEMBL8550946 0.73 ADORA2A (0.41) TDO2GAAADORA2A
SCHEMBL8546655 0.72 MAPK1 (0.42) ENPP1CYP2A6CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed