SCHEMBL8551565

SCHEMBL8551565

Clc1ccc(-c2nnc(Cl)c3c(Br)cccc23)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.42
MEN1 O00255 4/20 0.42
CYP1A2 P05177 3/20 0.42
CYP2C9 P11712 3/20 0.42
CYP2C19 P33261 3/20 0.42
ALDH1A1 P00352 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
HPGD P15428 2/20 0.40
ENPP3 O14638 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
KDR P35968 3/20 0.36
LMNA P02545 2/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 1/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549262 0.89 ALDH1A1 (0.41) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8551877 0.88 ESR1 (0.37) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8552712 0.79 ENPP1 (0.38) CYP2C9CYP2C19CYP3A4GAAADORA2A
SCHEMBL8549556 0.78 PLAU (0.44) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8546655 0.77 MAPK1 (0.42) KMT2ACYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL8549331 0.76 HSD11B1 (0.42) KMT2ACYP1A2ALDH1A1HPGDNPC1
SCHEMBL8549550 0.76 KDR (0.44) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL31359722 0.75 KMT2A (0.57) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL1396090 0.75 KMT2A (0.57) KMT2AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8553016 0.74 NPSR1 (0.45) KMT2AMEN1ALDH1A1NPSR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed