SCHEMBL8552929

SCHEMBL8552929

COC(=O)C=Cc1cnc[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 1.00
MEN1 O00255 2/20 1.00
KDM4E B2RXH2 5/20 0.64
BLM P54132 1/20 0.64
NPSR1 Q6W5P4 1/20 0.64
CYP3A4 P08684 1/20 0.64
TSHR P16473 1/20 0.64
SMYD3 Q9H7B4 1/20 0.44
AOC1 P19801 2/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
TYR P14679 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21334959 1.00 KMT2A (1.00) KMT2AMEN1KDM4EBLMNPSR1
SCHEMBL11598556 0.82 MEN1 (0.69) KMT2AMEN1KDM4EBLMNPSR1
SCHEMBL2567149 0.82 MEN1 (0.69) KMT2AMEN1KDM4EBLMNPSR1
Cis-Urocanic Acid SCHEMBL338885 0.78 CYP3A4 (1.00) KMT2AMEN1KDM4EBLMNPSR1
Cis-Urocanic Acid SCHEMBL1136889 0.78 CYP3A4 (1.00) KMT2AMEN1KDM4EBLMNPSR1
Cis-Urocanic Acid SCHEMBL12963908 0.78 CYP3A4 (1.00) KMT2AMEN1KDM4EBLMNPSR1
SCHEMBL23749602 0.77 CYP3A4 (0.70) KMT2AMEN1KDM4EBLMNPSR1
SCHEMBL15668642 0.77 CYP3A4 (0.70) KMT2AMEN1KDM4EBLMNPSR1
SCHEMBL25101013 0.76 KDM4E (0.64) KMT2AMEN1KDM4EBLMNPSR1
SCHEMBL22392209 0.74 MEN1 (0.58) KMT2AMEN1KDM4EBLMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed