Bromide

Bromide

SCHEMBL8553025

Br.COC(=O)COc1ccc(NC(=O)c2sc(C3CCNCC3)nc2C)cc1

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.49
KDM4E B2RXH2 1/20 0.49
KMT2A Q03164 6/20 0.46
MEN1 O00255 5/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.42
HPGD P15428 1/20 0.42
POLB P06746 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8554224 0.91 MAPT (0.50) MAPTKDM4EKMT2AMEN1ALDH1A1
SCHEMBL8554053 0.90 MAPT (0.51) MAPTKDM4EKMT2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL8592052 0.90 MAPT (0.50) MAPTKDM4EKMT2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL8593690 0.88 CXCR1 (0.44) MAPTKDM4EKMT2AMEN1ALDH1A1
Bromide SCHEMBL8553387 0.87 POLB (0.50) MAPTKDM4EKMT2AMEN1ALDH1A1
Bromide SCHEMBL8554165 0.85 KMT2A (0.42) MAPTKDM4EKMT2AMEN1ALDH1A1
Bromide SCHEMBL8551319 0.83 POLB (0.44) KMT2AMEN1ALDH1A1L3MBTL1HPGD
Bromide SCHEMBL8552807 0.81 MAPT (0.49) MAPTKDM4EKMT2AMEN1ALDH1A1
Bromide SCHEMBL8554391 0.78 LMNA (0.48) MAPTKDM4EKMT2AMEN1ALDH1A1
SCHEMBL8550534 0.78 KMT2A (0.44) MAPTKMT2AMEN1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858457-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM Dr. Karl Thomae GmbH (DE) 1998-08-19 EP disclosed
WO-1997015567-A1 5-MEMBERED HETEROCYCLES, PHARMACEUTICAL AGENTS CONTAINING SAID COMPOUNDS AND THE USE THEREOF AND METHODS OF PRODUCING THEM DR. KARL THOMAE GMBH (DE) 1997-05-01 WO disclosed