SCHEMBL8553397

SCHEMBL8553397

COc1ccc(-c2nc(Cc3ccccc3)oc2NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
KMT2A Q03164 1/20 0.49
GGT1 P19440 1/20 0.49
MAPT P10636 5/20 0.49
LMNA P02545 3/20 0.48
TP53 P04637 1/20 0.48
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
PTPN2 P17706 2/20 0.45
PTPN1 P18031 2/20 0.45
PTPN5 P54829 2/20 0.45
POLB P06746 2/20 0.44
LIMK2 P53671 2/20 0.44
HTT P42858 1/20 0.43
SLC40A1 Q9NP59 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026442 0.92 ALDH1A1 (0.46) ALDH1A1KMT2AGGT1MAPTLMNA
SCHEMBL8556104 0.90 ALDH1A1 (0.48) ALDH1A1KMT2AGGT1MAPTLMNA
SCHEMBL8556764 0.89 MAPT (0.54) ALDH1A1KMT2AMAPTLMNACYP2C9
SCHEMBL8556290 0.89 MAPT (0.51) ALDH1A1GGT1MAPTLMNATP53
SCHEMBL8560530 0.88 MAPT (0.52) ALDH1A1KMT2AMAPTLMNACYP3A4
SCHEMBL8559957 0.86 MAPT (0.47) ALDH1A1KMT2AMAPTLMNATP53
SCHEMBL8555221 0.85 MAPT (0.56) ALDH1A1KMT2AMAPTLMNAPTPN2
SCHEMBL8557761 0.85 MAPT (0.49) ALDH1A1KMT2AMAPTLMNAPTPN2
SCHEMBL8560689 0.85 ALDH1A1 (0.45) ALDH1A1KMT2AGGT1MAPTLMNA
SCHEMBL8557661 0.85 ALDH1A1 (0.45) ALDH1A1GGT1MAPTLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719163-A ARTHRITIS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed