SCHEMBL8553709

SCHEMBL8553709

Cc1ccc(-c2nnc(NC(=N)N)c3c(C#N)cccc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
KDR P35968 3/20 0.42
MAPT P10636 2/20 0.40
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 4/20 0.40
HPGD P15428 1/20 0.39
ENPP3 O14638 2/20 0.37
ERBB2 P04626 1/20 0.34
HTT P42858 2/20 0.34
ADORA1 P30542 2/20 0.34
ADORA2A P29274 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
F9 P00740 2/20 0.34
TP53 P04637 1/20 0.33
THRB P10828 1/20 0.33
F10 P00742 1/20 0.33
F11 P03951 1/20 0.33
F7 P08709 1/20 0.33
LMNA P02545 1/20 0.33
ADORA2B P29275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552217 0.90 KDM4E (0.37) ALDH1A1KDRMAPTGAANPSR1
SCHEMBL8548358 0.82 ALDH1A1 (0.46) ALDH1A1KDRMAPTGAANPSR1
SCHEMBL8547661 0.80 ALDH1A1 (0.43) ALDH1A1KDRMAPTGAANPSR1
SCHEMBL8547920 0.79 ALDH1A1 (0.64) ALDH1A1KDRMAPTGAANPSR1
SCHEMBL8552276 0.78 KDR (0.43) ALDH1A1KDRMAPTGAANPSR1
SCHEMBL8553714 0.77 PLAU (0.37) ALDH1A1KDRMAPTGAANPSR1
SCHEMBL8551333 0.75 ALDH1A1 (0.41) ALDH1A1MAPTGAANPSR1HPGD
Hydrochloric Acid SCHEMBL8551921 0.73 ALDH1A1 (0.46) ALDH1A1KDRMAPTGAANPSR1
SCHEMBL8374822 0.71 NPSR1 (0.39) ALDH1A1KDRMAPTGAANPSR1
SCHEMBL8518196 0.71 NPSR1 (0.39) ALDH1A1KDRMAPTGAANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed