SCHEMBL8553821

SCHEMBL8553821

Cc1c(OC(=O)O)nc2c(=O)[nH]c3ccccc3n12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
G6PD P11413 1/20 0.49
PKM P14618 1/20 0.49
HPGD P15428 1/20 0.49
ALOX12 P18054 1/20 0.49
HKDC1 Q2TB90 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
ADORA3 P0DMS8 12/20 0.47
ADORA1 P30542 3/20 0.47
ADORA2A P29274 2/20 0.47
NPSR1 Q6W5P4 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
PDE2A O00408 1/20 0.43
PDE6D O43924 1/20 0.43
PDE8A O60658 1/20 0.43
PDE5A O76074 1/20 0.43
PDE9A O76083 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557227 0.86 ADORA3 (0.54) POLBKDM4EALDH1A1MAPTG6PD
SCHEMBL8557884 0.84 ADORA3 (0.49) POLBKDM4EALDH1A1MAPTG6PD
SCHEMBL8555309 0.84 ADORA3 (0.47) POLBKDM4EALDH1A1MAPTG6PD
SCHEMBL8559120 0.83 ADORA3 (0.50) ADORA3PDE5APDE9A
SCHEMBL8557815 0.83 DAO (0.39) KDM4EALDH1A1HPGDTDP1ADORA3
SCHEMBL8557555 0.83 PDE5A (0.45) ADORA3PDE5APDE9A
SCHEMBL8557905 0.82 GRIN2D (0.43) ADORA3
SCHEMBL8558977 0.82 PDE5A (0.38) ADORA3PDE5APDE9A
SCHEMBL8557418 0.81 PDE5A (0.49) ALDH1A1MAPTHPGDALOX12ADORA3
SCHEMBL8553450 0.81 GRIA1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691970-B1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AG (DE) 1998-11-11 EP disclosed