SCHEMBL8553882

SCHEMBL8553882

Cc1cc(-c2nnn(C)n2)cc(C)c1OCCCC(=O)Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 5/20 0.37
FFAR1 O14842 3/20 0.37
FFAR4 Q5NUL3 2/20 0.36
CYP3A4 P08684 1/20 0.36
KCNH2 Q12809 1/20 0.36
CACNA1C Q13936 1/20 0.36
SCN5A Q14524 1/20 0.36
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
HDAC3 O15379 1/20 0.35
NCOR1 O75376 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
MMP1 P03956 1/20 0.34
MMP9 P14780 1/20 0.34
MMP8 P22894 1/20 0.34
TP53 P04637 1/20 0.34
CYP2C8 P10632 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551826 0.89 FFAR4 (0.44) HDAC6FFAR1FFAR4CYP3A4KCNH2
SCHEMBL8604570 0.89 HDAC6 (0.38) HDAC6FFAR1FFAR4CYP3A4KCNH2
SCHEMBL9091116 0.87 TSHR (0.43) HDAC6HDAC3NCOR1HDAC1HDAC2
SCHEMBL9089363 0.86 NPSR1 (0.42) HDAC6THRATHRBALDH1A1MEN1
SCHEMBL8824429 0.83 THRA (0.39) HDAC6THRATHRBHDAC3NCOR1
SCHEMBL9089935 0.81 HDAC6 (0.39) HDAC6HDAC3NCOR1HDAC1HDAC2
SCHEMBL8557288 0.81 HDAC6 (0.39) HDAC6HDAC3NCOR1HDAC1HDAC2
SCHEMBL9089670 0.81 RAB9A (0.40) HDAC6HDAC3NCOR1HDAC1HDAC2
SCHEMBL8553780 0.81 NPC1 (0.36) HDAC6FFAR1CYP3A4NPC1NFKB1
SCHEMBL8661865 0.80 NPC1 (0.34) HDAC6FFAR1CYP3A4TP53NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846986-A Therapeutic phenoxyalkylazoles and phenoxyalkylazines SANOFI (FR) 1998-12-08 US disclosed
US-5721261-A TREATING PICORNAVIRUS INFECTIONS SANOFI PHARMACEUTICALS, INC. (US) 1998-02-24 US disclosed
US-5552420-A TREATING PICORNAVIRAL INFECTIONS STERLING WINTHROP INC. (US) 1996-09-03 US disclosed
WO-1995031452-A1 THERAPEUTIC PHENOXYALKYLAZOLES AND PHENOXYALKYLAZINES SANOFI WINTHROP, INC. (US) 1995-11-23 WO disclosed