SCHEMBL8553953

SCHEMBL8553953

CCCCc1ccc(CC(CC(N)=O)NCCC)cc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PLK1 P53350 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
S1PR2 O95136 1/20 0.41
S1PR1 P21453 1/20 0.41
POLB P06746 1/20 0.40
F13A1 P00488 1/20 0.40
TGM2 P21980 1/20 0.40
RARB P10826 1/20 0.40
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6803279 1.00 SIGMAR1 (0.45) SIGMAR1NPC1RAB9ASMN1; SMN2PLK1
SCHEMBL6801926 0.94 SIGMAR1 (0.48) SIGMAR1NPC1RAB9ASMN1; SMN2PLK1
SCHEMBL6800799 0.89 SIGMAR1 (0.49) SIGMAR1S1PR2S1PR1THRATHRB
SCHEMBL27347413 0.86 LOXL2 (0.38) SIGMAR1
SCHEMBL6796677 0.86 HPGD (0.40) SIGMAR1SMN1; SMN2ALDH1A1HPGD
Hydrochloric Acid SCHEMBL3059803 0.83 SIGMAR1 (0.51) SIGMAR1NPC1RAB9APOLB
SCHEMBL6802210 0.78 AKR1C3 (0.42) SIGMAR1
SCHEMBL6803232 0.78 ALDH1A1 (0.49) NPC1RAB9ASMN1; SMN2PLK1ALDH1A1
SCHEMBL6802810 0.77 HTR2A (0.46) SIGMAR1
Hydrochloric Acid SCHEMBL6807729 0.77 S1PR1 (0.51) NPC1RAB9ASMN1; SMN2PLK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0854863-A1 ESTERS AND AMIDES AS PLA2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-07-29 EP disclosed
WO-1997003951-A1 ESTERS AND AMIDES AS PLA2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-02-06 WO disclosed