SCHEMBL8554583

SCHEMBL8554583

CC(C)=CCOc1ccc(C)c2c1C(C)(C)C(=O)N2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.37
MTNR1A P48039 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
TRPA1 O75762 1/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
PTGES O14684 4/20 0.36
MMP1 P03956 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34
MMP12 P39900 1/20 0.34
PTGS1 P23219 2/20 0.34
PTGS2 P35354 2/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8555134 0.84 ALDH1A1 (0.37) PDE4BKDM4EALDH1A1CYP3A4HPGD
SCHEMBL8557018 0.83 PDK2 (0.33) ALDH1A1
SCHEMBL8557014 0.83 PDK2 (0.33) ALDH1A1
SCHEMBL8559248 0.83 ALDH1A1 (0.42) PDE4BKDM4EALDH1A1HPGD
SCHEMBL8596431 0.83 KMT2A (0.32) ALDH1A1PTPN1
SCHEMBL8596432 0.83 KMT2A (0.32) ALDH1A1PTPN1
SCHEMBL8555928 0.82 PDK2 (0.35)
SCHEMBL8557766 0.81 PDK2 (0.32) ALDH1A1
SCHEMBL8557765 0.81 PDK2 (0.32) ALDH1A1
SCHEMBL6582041 0.77 PDK2 (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653426-B1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA CO (JP) 1998-07-22 EP disclosed
US-5510366-A INOTROPIC, ANTIARRHYMTHMIA AGENTS, VASODILATORS KOWA CO., LTD. (JP) 1996-04-23 US disclosed
EP-0653426-A1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA COMPANY, LTD. (JP) 1995-05-17 EP disclosed