SCHEMBL8554657

SCHEMBL8554657

CS(=O)(=O)CCC(Cc1ccccc1C(N)=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.38
AURKA O14965 3/20 0.37
RPS6KB1 P23443 3/20 0.37
SLC6A4 P31645 6/20 0.36
SLC6A2 P23975 5/20 0.36
SLC6A3 Q01959 5/20 0.36
CYP3A4 P08684 3/20 0.36
CYP2D6 P10635 3/20 0.36
TNF P01375 1/20 0.36
PTPRG P23470 1/20 0.36
CNR1 P21554 1/20 0.36
MAPK14 Q16539 1/20 0.36
KCNH2 Q12809 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308083 0.85 CYP2D6 (0.48) SLC6A4SLC6A2SLC6A3CYP3A4CYP2D6
SCHEMBL8597114 0.85 IKBKB (0.39) RPS6KB1CYP2D6IKBKB
SCHEMBL4468913 0.78 TNF (0.44) SLC6A4SLC6A2SLC6A3CYP3A4CYP2D6
SCHEMBL8390128 0.74 NOTUM (0.35) MAPTRAB9A
SCHEMBL8554659 0.72 HPGD (0.45) SLC6A4SLC6A2SLC6A3CYP3A4CYP2D6
SCHEMBL6425161 0.71 TACR2 (0.65) TACR2
SCHEMBL4468917 0.71 SLC6A2 (0.50) SLC6A4SLC6A2SLC6A3CYP3A4CYP2D6
SCHEMBL16649632 0.70 SLC6A2 (0.43) SLC6A4SLC6A2SLC6A3CYP3A4CYP2D6
SCHEMBL4564260 0.69 IKBKB (0.52) SLC6A3CYP3A4MAPTIKBKB
SCHEMBL4468911 0.68 SLC6A2 (0.38) SLC6A4SLC6A2SLC6A3CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0882038-A1 NOVEL SUBSTITUTED N-METHYL-N-(4-(PIPERIDIN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES HOECHST MARION ROUSSEL, INC. (US) 1998-12-09 EP disclosed
WO-1997030990-A1 NOVEL SUBSTITUTED N-METHYL-N-(4-(PIPERIDIN-1-YL)-2-(ARYL)BUTYL)BENZAMIDES USEFUL FOR THE TREATMENT OF ALLERGIC DISEASES HOECHST MARION ROUSSEL, INC. (US) 1997-08-28 WO disclosed