SCHEMBL4468911

SCHEMBL4468911

CS(=O)(=O)CC[C@H](CNC=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 14/20 0.38
SLC6A4 P31645 14/20 0.38
SLC6A3 Q01959 14/20 0.38
CYP3A4 P08684 12/20 0.37
CYP2D6 P10635 12/20 0.37
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KCNH2 Q12809 9/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4468917 0.85 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL6770900 0.81 SLC6A4 (0.44) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL4475059 0.81 ALDH1A1 (0.38) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL6770174 0.80 SLC6A4 (0.47) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL4471202 0.77 ALDH1A1 (0.37) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL8554659 0.76 HPGD (0.45) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL4468913 0.75 TNF (0.44) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL6770082 0.74 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL16649632 0.73 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL6769279 0.72 SIGMAR1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7592344-B2 NK1 and NK2-antagonists and compositions and methods of using the same SOLVAY PHARMACEUTICALS GMBH (DE) 2009-09-22 US disclosed
EP-1954678-A1 NOVEL NK1 AND NK2 ANTAGONISTS Solvay Pharmaceuticals GmbH (DE) 2008-08-13 EP disclosed
US-20070149537-A1 NK1 and NK2-antagonists and compositions and methods of using the same SOLVAY PHARMACEUTICALS GMBH (DE) 2007-06-28 US disclosed
WO-2007063086-A1 NOVEL NK1 AND NK2 ANTAGONISTS SOLVAY PHARMACEUTICALS GMBH (DE) 2007-06-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070149537-A1 NK1 and NK2-antagonists and compositions and methods of using the same HRH2, PROKR2, BDKRB2 SLC6A2 1388/4885SLC6A4 2566/4885SLC6A3 2380/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.