SCHEMBL8554739

SCHEMBL8554739

O=C1C(Br)CCN1c1ccc(F)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.45
DRD3 P35462 2/20 0.45
ALDH1A1 P00352 2/20 0.43
HSP90AA1 P07900 1/20 0.43
KCNH2 Q12809 1/20 0.43
KAT2B Q92831 2/20 0.42
PIN1 Q13526 1/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
GAA P10253 2/20 0.42
RAD51 Q06609 1/20 0.40
SLC6A2 P23975 3/20 0.40
SLC6A4 P31645 3/20 0.40
SLC6A3 Q01959 2/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18740427 0.88 RAD51 (0.41) KCNH2CYP2D6RAD51SLC6A2SLC6A4
SCHEMBL8554615 0.82 SLC6A2 (0.47) DRD2DRD3ALDH1A1HSP90AA1KCNH2
SCHEMBL22481515 0.81 HDAC6 (0.46) ROCK2HDAC6LMNA
SCHEMBL18740192 0.80 ROCK2 (0.38) KMT2AMEN1SLC6A2SLC6A4SLC6A3
SCHEMBL16874727 0.79 CCR1 (0.39) ALDH1A1CYP1A2CYP2C19MAPTROCK2
SCHEMBL16885989 0.79 CCR1 (0.39) ALDH1A1CYP1A2CYP2C19MAPTROCK2
SCHEMBL6530315 0.79 CYP2D6 (0.50) DRD2DRD3KCNH2CYP1A2CYP2D6
SCHEMBL2289335 0.79 ALDH1A1 (0.46) DRD2DRD3ALDH1A1HSP90AA1KCNH2
SCHEMBL27509176 0.79 DRD2 (0.40) DRD2DRD3ALDH1A1HSP90AA1KCNH2
SCHEMBL5827625 0.77 MCHR1 (0.47) ALDH1A1SLC6A2SLC6A4SLC6A3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1203599-A Substitued pyrrolidinone, thiazolidinone or oxazolidinone as herbicides ZENECA LTD (GB) 1998-12-30 CN disclosed
EP-0863894-A1 SUBSTITUTED PYRROLIDINONE, THIAZOLIDINONE OR OXAZOLIDINONE AS HERBICIDES ZENECA LIMITED (GB) 1998-09-16 EP disclosed
US-5705456-A AZETIDIN-2-ONES ZENECA LIMITED (GB) 1998-01-06 US disclosed
WO-1997020838-A1 SUBSTITUTED PYRROLIDINONE, THIAZOLIDINONE OR OXAZOLIDINONE AS HERBICIDES ZENECA LIMITED (GB) 1997-06-12 WO disclosed