SCHEMBL8554918

SCHEMBL8554918

[CH2]c1cccc(C(=O)Nc2ccc(C)cn2)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.71
RAB9A P51151 11/20 0.61
L3MBTL1 Q9Y468 1/20 0.58
KDM4E B2RXH2 2/20 0.58
NPC1 O15118 8/20 0.56
POLB P06746 1/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
RXFP1 Q9HBX9 1/20 0.56
TDP1 Q9NUW8 1/20 0.55
MAPT P10636 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.52
TP53 P04637 2/20 0.52
PKM P14618 2/20 0.52
GLA P06280 1/20 0.52
GAA P10253 1/20 0.52
HSD17B10 Q99714 1/20 0.52
TSHR P16473 2/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554924 0.87 ALDH1A1 (0.77) ALDH1A1RAB9AL3MBTL1KDM4ENPC1
SCHEMBL14758512 0.83 RAB9A (0.71) ALDH1A1RAB9AL3MBTL1KDM4ENPC1
SCHEMBL26758744 0.82 ALDH1A1 (0.70) ALDH1A1RAB9AL3MBTL1KDM4ENPC1
SCHEMBL3529609 0.82 KDM4E (0.72) ALDH1A1RAB9AKDM4ENPC1POLB
SCHEMBL8555107 0.81 NPC1 (0.65) ALDH1A1RAB9AKDM4ENPC1POLB
SCHEMBL21709858 0.79 KDM4E (0.82) ALDH1A1RAB9AL3MBTL1KDM4ENPC1
SCHEMBL30216783 0.79 KDM4E (0.82) ALDH1A1RAB9AL3MBTL1KDM4ENPC1
SCHEMBL7348632 0.78 RAB9A (0.66) ALDH1A1RAB9AL3MBTL1KDM4ENPC1
SCHEMBL1196619 0.78 NPC1 (0.65) RAB9AL3MBTL1KDM4ENPC1POLB
SCHEMBL14979240 0.78 DEGS1 (0.73) ALDH1A1RAB9AKDM4ENPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP claimed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US claimed
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP disclosed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US disclosed