SCHEMBL8555054

SCHEMBL8555054

COc1cc(Cc2nccc3ccccc23)cc(OC)c1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 5/20 0.56
SMN1; SMN2 Q16637 5/20 0.56
PDE3A Q14432 5/20 0.56
CYP3A4 P08684 4/20 0.56
MAPK1 P28482 4/20 0.56
PDE3B Q13370 4/20 0.56
LMNA P02545 3/20 0.56
USP2 O75604 2/20 0.56
ALDH1A1 P00352 2/20 0.56
HIF1A Q16665 2/20 0.56
RAB9A P51151 2/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2C9 P11712 2/20 0.56
TSHR P16473 2/20 0.56
PDE4A P27815 2/20 0.56
KCNH2 Q12809 2/20 0.56
PDE4D Q08499 2/20 0.56
PDE2A O00408 1/20 0.56
ABCC4 O15439 1/20 0.56
PDE5A O76074 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4429531 0.86 PDE10A (0.75) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1
SCHEMBL23457662 0.84 PDE10A (0.77) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1
SCHEMBL8554954 0.83 PDE10A (0.53) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1
Hydrochloric Acid SCHEMBL10677574 0.80 PDE10A (0.61) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1
SCHEMBL149392 0.80 PDE10A (0.55) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1
SCHEMBL10867414 0.80 RAB9A (0.58) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1
SCHEMBL1445588 0.78 PDE10A (0.66) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1
SCHEMBL8559774 0.78 RAB9A (0.56) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1
SCHEMBL192576 0.78 TUBB4A (0.46) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1
SCHEMBL1445506 0.78 PDE10A (0.53) PDE10ASMN1; SMN2PDE3ACYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0617022-B1 6,7, dialkoxy-3,4-dihydroisoquinolin-8-ol, process for preparation thereof and process for preparation of 6,7-dialkoxy-1,2,3,4-tetrahydroisoquinolin-8-ol using the compound BANYU PHARMA CO LTD (JP) 1998-02-11 EP disclosed
EP-0617022-A1 6,7, dialkoxy-3,4-dihydroisoquinolin-8-ol, process for preparation thereof and process for preparation of 6,7-dialkoxy-1,2,3,4-tetrahydroisoquinolin-8-ol using the compound BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-09-28 EP disclosed