SCHEMBL8554954

SCHEMBL8554954

COc1cc(Cc2nccc3ccccc23)cc(OC)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.53
PDE3A Q14432 4/20 0.53
PDE3B Q13370 3/20 0.53
CYP3A4 P08684 4/20 0.48
MAPK1 P28482 4/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
LMNA P02545 3/20 0.48
USP2 O75604 2/20 0.48
ALDH1A1 P00352 2/20 0.48
HIF1A Q16665 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C9 P11712 2/20 0.48
TSHR P16473 2/20 0.48
PDE4A P27815 2/20 0.48
KCNH2 Q12809 2/20 0.48
RAB9A P51151 2/20 0.48
PDE4D Q08499 2/20 0.48
PDE2A O00408 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1445580 0.89 PDE10A (0.51) PDE10APDE3APDE3BCYP3A4MAPK1
SCHEMBL1445588 0.87 PDE10A (0.66) PDE10APDE3APDE3BCYP3A4MAPK1
Water SCHEMBL28228890 0.85 PDE10A (0.64) PDE10APDE3APDE3BCYP3A4MAPK1
SCHEMBL8555054 0.83 PDE10A (0.56) PDE10APDE3APDE3BCYP3A4MAPK1
SCHEMBL4429531 0.80 PDE10A (0.75) PDE10APDE3APDE3BCYP3A4MAPK1
SCHEMBL8554309 0.78 PDE10A (0.56) PDE10APDE3APDE3BCYP3A4MAPK1
SCHEMBL12402267 0.78 PDE10A (0.48) PDE10APDE3APDE3BCYP3A4MAPK1
SCHEMBL29373118 0.77 ACHE (0.49) PDE10APDE3APDE3BCYP3A4MAPK1
SCHEMBL232662 0.77 ACHE (0.49) PDE10APDE3APDE3BCYP3A4MAPK1
SCHEMBL23457928 0.77 RAB9A (0.50) PDE10APDE3APDE3BMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0617022-B1 6,7, dialkoxy-3,4-dihydroisoquinolin-8-ol, process for preparation thereof and process for preparation of 6,7-dialkoxy-1,2,3,4-tetrahydroisoquinolin-8-ol using the compound BANYU PHARMA CO LTD (JP) 1998-02-11 EP disclosed
EP-0617022-A1 6,7, dialkoxy-3,4-dihydroisoquinolin-8-ol, process for preparation thereof and process for preparation of 6,7-dialkoxy-1,2,3,4-tetrahydroisoquinolin-8-ol using the compound BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-09-28 EP disclosed