SCHEMBL8555936

SCHEMBL8555936

Cc1cccc([CH]Cc2ccncc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.44
TP53 P04637 1/20 0.44
NPC1 O15118 2/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
GAA P10253 1/20 0.42
RAB9A P51151 1/20 0.42
PKM P14618 2/20 0.40
KDM4E B2RXH2 2/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
CHEK1 O14757 1/20 0.39
CDK1 P06493 1/20 0.39
CDK4 P11802 1/20 0.39
CCNA2 P20248 1/20 0.39
CCND1 P24385 1/20 0.39
CDK2 P24941 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4953933 0.84 TP53 (0.48) TDP1TP53NPC1CASP3SENP8
SCHEMBL8207446 0.84 TP53 (0.48) TDP1TP53NPC1CASP3SENP8
SCHEMBL7377625 0.82 VNN1 (0.45) TDP1TP53KDM4ELMNAHPGD
SCHEMBL8097032 0.82 TP53 (0.50) TDP1TP53NPC1CASP3SENP8
SCHEMBL16494233 0.79 TP53 (0.44) TDP1TP53NPC1CASP3SENP8
SCHEMBL5966235 0.77 CYP1A2 (0.46) LMNACYP1A2MAOBSMN1; SMN2CYP11B1
SCHEMBL8202649 0.75 CYP3A4 (0.48) NPC1RAB9AKDM4ELMNAHPGD
SCHEMBL1611151 0.73 TP53 (0.58) TDP1TP53NPC1CASP3SENP8
SCHEMBL8200491 0.73 CYP11B2 (0.47) NPC1RAB9AKDM4EKMT2ACYP1A2
SCHEMBL8667992 0.72 RELA (0.43) NPC1RAB9AKDM4ECHEK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832076-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-04-01 EP disclosed