SCHEMBL8555953

SCHEMBL8555953

CCC(=O)c1[nH]c2cc(C(=O)NCc3ccccc3Cl)ccc2c1C(=O)C(C)C

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 6/20 0.56
SMN1; SMN2 Q16637 5/20 0.52
CASP6 P55212 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.46
MAPK1 P28482 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPK3 P27361 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
LMNA P02545 2/20 0.45
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.44
PKM P14618 1/20 0.44
HTT P42858 1/20 0.44
HTR3A P46098 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18073895 0.85 ROCK2 (0.56) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK1
SCHEMBL8555308 0.79 ROCK2 (0.62) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK1
SCHEMBL8555167 0.78 ROCK2 (0.63) ROCK2SMN1; SMN2CASP6MAPK1ALDH1A1
SCHEMBL8556569 0.78 ROCK2 (0.63) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK1
SCHEMBL7707825 0.77 ROCK2 (0.57) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK1
SCHEMBL8554376 0.76 ROCK2 (0.56) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK1
SCHEMBL8556812 0.75 ROCK2 (0.60) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK1
SCHEMBL7701986 0.74 ROCK2 (0.54) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK1
SCHEMBL8629096 0.72 MAPT (0.55) ALDH1A1CYP3A4CYP2C19LMNAKDM4E
SCHEMBL17783613 0.72 ROCK2 (1.00) ROCK2SMN1; SMN2CASP6MAPK1MAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820441-A1 INDOLE DERIVATIVES AS cGMP-PDE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-01-28 EP disclosed