SCHEMBL8556812

SCHEMBL8556812

CCCc1[nH]c2cc(C(=O)NCc3ccccc3Cl)ccc2c1Cl

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 7/20 0.60
SMN1; SMN2 Q16637 4/20 0.56
CASP6 P55212 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.53
MAPK3 P27361 1/20 0.49
MAPK1 P28482 1/20 0.49
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
POLB P06746 1/20 0.48
ROCK1 Q13464 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7707825 0.89 ROCK2 (0.57) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK3
SCHEMBL8554376 0.88 ROCK2 (0.56) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK3
SCHEMBL18073895 0.87 ROCK2 (0.56) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK3
SCHEMBL7701986 0.85 ROCK2 (0.54) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK3
SCHEMBL8555308 0.81 ROCK2 (0.62) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK3
SCHEMBL7707256 0.79 KMT2A (0.46) ROCK2SMN1; SMN2CASP6KDM4ETP53
SCHEMBL8556569 0.77 ROCK2 (0.63) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK3
SCHEMBL8555167 0.77 ROCK2 (0.63) ROCK2SMN1; SMN2CASP6MAPK3MAPK1
SCHEMBL17783613 0.75 ROCK2 (1.00) ROCK2SMN1; SMN2CASP6MAPK3MAPK1
SCHEMBL8555953 0.75 ROCK2 (0.56) ROCK2SMN1; SMN2CASP6L3MBTL1MAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820441-A1 INDOLE DERIVATIVES AS cGMP-PDE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-01-28 EP disclosed