SCHEMBL8556040

SCHEMBL8556040

Cc1cc(-c2nnn(C)n2)cc(C)c1OCCCc1nc(CCl)co1

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553973 0.87 NR1I2 (0.41) NR1I2CYP3A4CYP2D6
SCHEMBL8555193 0.79 NR1I2 (0.41) NR1I2CYP3A4CYP2D6
SCHEMBL8552034 0.78 NR1I2 (0.35) NR1I2CYP3A4CYP2D6
SCHEMBL8603712 0.78 NR1I2 (0.37) NR1I2CYP3A4CYP2D6
SCHEMBL9078729 0.74 RAB9A (0.41) NR1I2CYP3A4CYP2D6
SCHEMBL8551728 0.74 NR1I2 (0.34) NR1I2CYP3A4CYP2D6
SCHEMBL8558294 0.74 NR1I2 (0.41) NR1I2CYP3A4CYP2D6
SCHEMBL8824410 0.74 NR1I2 (0.35) NR1I2CYP3A4CYP2D6
SCHEMBL8824405 0.74 NPC1 (0.34) NR1I2CYP3A4CYP2D6
SCHEMBL8553780 0.74 NPC1 (0.36) NR1I2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5846986-A Therapeutic phenoxyalkylazoles and phenoxyalkylazines SANOFI (FR) 1998-12-08 US disclosed
US-5721261-A TREATING PICORNAVIRUS INFECTIONS SANOFI PHARMACEUTICALS, INC. (US) 1998-02-24 US disclosed
US-5552420-A TREATING PICORNAVIRAL INFECTIONS STERLING WINTHROP INC. (US) 1996-09-03 US disclosed
WO-1995031452-A1 THERAPEUTIC PHENOXYALKYLAZOLES AND PHENOXYALKYLAZINES SANOFI WINTHROP, INC. (US) 1995-11-23 WO disclosed