SCHEMBL8556339

SCHEMBL8556339

CC(=O)C1(c2ccccc2)CCN(CCCC2CC(c3ccc(Cl)c(Cl)c3)CN(Cc3ccccc3)C2=O)CC1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.58
TACR2 P21452 10/20 0.58
TACR3 P29371 6/20 0.58
HTR7 P34969 1/20 0.41
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
KCNA3 P22001 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8594002 0.83 TACR1 (0.46) TACR1TACR2TACR3ADRA2AADRA2B
Hydrochloric Acid SCHEMBL8368423 0.83 TACR1 (0.53) TACR1TACR2TACR3
SCHEMBL8559945 0.80 TACR2 (0.60) TACR1TACR2TACR3HTR7
SCHEMBL8558380 0.79 HPGD (0.40) TACR1TACR2
SCHEMBL8559948 0.76 TACR2 (0.55) TACR1TACR2TACR3HTR7ADRA2A
Hydrochloric Acid SCHEMBL8593049 0.75 CCR3 (0.42) TACR1MEN1KMT2A
SCHEMBL8556923 0.74 TACR2 (0.58) TACR1TACR2TACR3ADRA2AADRA2B
SCHEMBL8561168 0.74 PDE4A (0.40) TACR1TACR2
SCHEMBL7844998 0.73 TACR1 (1.00) TACR1TACR2TACR3
Hydrochloric Acid SCHEMBL8368100 0.72 TACR2 (0.47) TACR1TACR2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807865-A 3,3-disubstituted piperidine derivatives and their use as therapeutic agents MERCK SHARP & DOHME LIMITED (GB) 1998-09-15 US disclosed