SCHEMBL8561168

SCHEMBL8561168

CS(=O)(=O)OCCCC1CC(c2ccc(Cl)c(Cl)c2)CN(Cc2ccccc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
KCNA5 P22460 1/20 0.35
TACR1 P25103 9/20 0.35
TACR2 P21452 7/20 0.35
SLC6A3 Q01959 4/20 0.35
SLC6A2 P23975 3/20 0.35
SLC6A4 P31645 3/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558380 0.83 HPGD (0.40) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL8558084 0.79 PTAFR (0.37) PDE4APDE4BPDE4CPDE4DTACR1
SCHEMBL8556339 0.74 TACR1 (0.58) TACR1TACR2
Hydrochloric Acid SCHEMBL8593049 0.73 CCR3 (0.42) TACR1SLC6A2SLC6A4
SCHEMBL8594002 0.72 TACR1 (0.46) TACR1TACR2
Hydrochloric Acid SCHEMBL8368423 0.71 TACR1 (0.53) TACR1TACR2POLB
SCHEMBL8556923 0.70 TACR2 (0.58) PDE4DTSHRTACR1TACR2SLC6A3
SCHEMBL8300797 0.67 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DKCNA5
SCHEMBL8564881 0.67 PDE4A (0.38) PDE4APDE4BPDE4CPDE4DHPGD
SCHEMBL7847578 0.67 TACR1 (0.61) TACR1TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807865-A 3,3-disubstituted piperidine derivatives and their use as therapeutic agents MERCK SHARP & DOHME LIMITED (GB) 1998-09-15 US disclosed