SCHEMBL8556923

SCHEMBL8556923

O=C1C(CCCN2CCC(n3c(=O)[nH]c4ccccc43)CC2)CC(c2ccc(Cl)c(Cl)c2)CN1Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 2/20 0.58
TACR1 P25103 2/20 0.58
TACR3 P29371 2/20 0.58
CCR5 P51681 2/20 0.58
OPRM1 P35372 11/20 0.56
OPRL1 P41146 5/20 0.53
OPRK1 P41145 3/20 0.53
CYP2D6 P10635 4/20 0.51
PMP22 Q01453 3/20 0.51
USP2 O75604 3/20 0.51
CYP1A2 P05177 3/20 0.51
MEN1 O00255 2/20 0.51
SLC22A2 O15244 2/20 0.51
GMNN O75496 2/20 0.51
LMNA P02545 2/20 0.51
ADRB2 P07550 2/20 0.51
ADRB1 P08588 2/20 0.51
CYP3A4 P08684 2/20 0.51
HTR1A P08908 2/20 0.51
ADRA2A P08913 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560042 0.81 TACR2 (0.62) TACR2TACR1TACR3CCR5OPRM1
Hydrochloric Acid SCHEMBL8593049 0.76 CCR3 (0.42) TACR1MEN1SLC6A2SLC6A4KMT2A
SCHEMBL8558380 0.75 HPGD (0.40) TACR2TACR1SLC6A2SLC6A4SLC6A3
SCHEMBL8556339 0.74 TACR1 (0.58) TACR2TACR1TACR3MEN1ADRA2A
SCHEMBL7842031 0.74 TACR1 (1.00) TACR2TACR1TACR3CCR5OPRM1
SCHEMBL24709114 0.72 CYP2D6 (0.74) OPRM1OPRL1OPRK1CYP2D6PMP22
SCHEMBL31000422 0.72 CYP2D6 (0.74) OPRM1OPRL1OPRK1CYP2D6PMP22
SCHEMBL3665096 0.72 OPRM1 (1.00) OPRM1OPRL1OPRK1CYP3A4DRD2
SCHEMBL5984495 0.72 CYP2D6 (0.85) OPRM1OPRL1OPRK1CYP2D6PMP22
SCHEMBL24708725 0.71 CHRM1 (0.73) OPRM1OPRL1OPRK1CYP2D6PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807865-A 3,3-disubstituted piperidine derivatives and their use as therapeutic agents MERCK SHARP & DOHME LIMITED (GB) 1998-09-15 US disclosed