SCHEMBL8558380

SCHEMBL8558380

O=C1C(CCCO)CC(c2ccc(Cl)c(Cl)c2)CN1Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
PDE4A P27815 3/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
SLC6A3 Q01959 3/20 0.38
KCNH2 Q12809 1/20 0.38
KCNA5 P22460 1/20 0.37
TACR1 P25103 3/20 0.37
LIPG Q9Y5X9 1/20 0.35
TACR2 P21452 1/20 0.35
SIGMAR1 Q99720 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561168 0.83 PDE4A (0.40) HPGDTSHRPDE4APDE4BPDE4C
SCHEMBL8558084 0.79 PTAFR (0.37) PDE4APDE4BPDE4CPDE4DTACR1
SCHEMBL8556339 0.79 TACR1 (0.58) TACR1TACR2
Hydrochloric Acid SCHEMBL8593049 0.79 CCR3 (0.42) SLC6A2SLC6A4TACR1
Hydrochloric Acid SCHEMBL8368423 0.79 TACR1 (0.53) TACR1TACR2SIGMAR1
SCHEMBL8556923 0.75 TACR2 (0.58) TSHRPDE4DSLC6A2SLC6A4SLC6A3
SCHEMBL8594002 0.75 TACR1 (0.46) TACR1TACR2SIGMAR1
SCHEMBL3646955 0.70 RORC (0.48) SLC6A2SLC6A4SLC6A3KCNH2SIGMAR1
SCHEMBL8564881 0.68 PDE4A (0.38) HPGDTSHRPDE4APDE4BPDE4C
SCHEMBL7846535 0.65 OPRK1 (0.43) SLC6A2SLC6A4SLC6A3KCNA5SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807865-A 3,3-disubstituted piperidine derivatives and their use as therapeutic agents MERCK SHARP & DOHME LIMITED (GB) 1998-09-15 US disclosed