SCHEMBL8556582

SCHEMBL8556582

Clc1ccc(C(c2ccccc2)N2CCN(c3ncsn3)CC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.61
NPSR1 Q6W5P4 1/20 0.61
CHRM2 P08172 3/20 0.56
ADRA2A P08913 3/20 0.56
ADRA1A P35348 3/20 0.56
DRD3 P35462 3/20 0.56
KCNH2 Q12809 3/20 0.56
HTR1A P08908 2/20 0.56
CHRM1 P11229 2/20 0.56
DRD1 P21728 2/20 0.56
TBXA2R P21731 2/20 0.56
SLC6A2 P23975 2/20 0.56
SLC6A4 P31645 2/20 0.56
SLC6A3 Q01959 2/20 0.56
BCL2 P10415 1/20 0.56
HRH3 Q9Y5N1 1/20 0.56
CYP2D6 P10635 2/20 0.55
TSHR P16473 2/20 0.55
CYP2C19 P33261 1/20 0.55
TDP1 Q9NUW8 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560914 0.80 KCNH2 (0.55) KDM4ENPSR1CHRM2ADRA2AADRA1A
SCHEMBL11396110 0.80 KDM4E (0.61) KDM4ENPSR1CHRM2ADRA2AADRA1A
SCHEMBL7668121 0.80 CHRM2 (0.83) KDM4ENPSR1CHRM2ADRA2AADRA1A
Chlorcyclizine SCHEMBL13724147 0.72 KCNH2 (1.00) KDM4ENPSR1CHRM2ADRA2AADRA1A
Chlorcyclizine SCHEMBL12157065 0.72 KCNH2 (1.00) KDM4ENPSR1CHRM2ADRA2AADRA1A
Chlorcyclizine SCHEMBL16769331 0.72 KCNH2 (1.00) KDM4ENPSR1CHRM2ADRA2AADRA1A
SCHEMBL1381608 0.72 DRD3 (0.66) KDM4ENPSR1CHRM2ADRA2AADRA1A
SCHEMBL13900811 0.72 KCNH2 (0.76) KDM4ENPSR1CHRM2ADRA2AADRA1A
SCHEMBL11212785 0.72 KCNH2 (0.71) KDM4ENPSR1CHRM2ADRA2AADRA1A
Chlorcyclizine SCHEMBL4383 0.72 KCNH2 (1.00) KDM4ENPSR1CHRM2ADRA2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883622-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1998-12-16 EP claimed
WO-1997031923-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1997-09-04 WO claimed
EP-0883606-A1 PROCESS FOR SCAVENGING THIOLS APOTEX INC. (CA) 1998-12-16 EP disclosed
WO-1997031893-A1 PROCESS FOR SCAVENGING THIOLS APOTEX INC. (CA) 1997-09-04 WO disclosed