SCHEMBL8560914

SCHEMBL8560914

Clc1ccc(C(c2ccccc2)N2CCN(Cc3ncsn3)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.55
HRH1 P35367 5/20 0.55
OPRK1 P41145 3/20 0.55
ADORA3 P0DMS8 2/20 0.55
CNR1 P21554 2/20 0.55
GHSR Q92847 2/20 0.55
LMNA P02545 2/20 0.55
NR1I2 O75469 1/20 0.55
PDE4D Q08499 1/20 0.55
DRD3 P35462 6/20 0.54
CHRM2 P08172 4/20 0.54
ADRA2A P08913 4/20 0.54
ADRA1A P35348 4/20 0.54
SLC6A2 P23975 4/20 0.54
SLC6A4 P31645 4/20 0.54
SLC6A3 Q01959 4/20 0.54
CYP2D6 P10635 3/20 0.54
CHRM1 P11229 3/20 0.54
DRD1 P21728 3/20 0.54
USP2 O75604 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556582 0.80 KDM4E (0.61) KCNH2HRH1OPRK1LMNADRD3
SCHEMBL588111 0.79 KCNH2 (0.78) KCNH2HRH1OPRK1ADORA3CNR1
SCHEMBL588110 0.79 KCNH2 (0.78) KCNH2HRH1OPRK1ADORA3CNR1
SCHEMBL3611802 0.79 KCNH2 (0.78) KCNH2HRH1OPRK1ADORA3CNR1
SCHEMBL12464946 0.79 KCNH2 (0.80) KCNH2HRH1OPRK1ADORA3CNR1
Hydrochloric Acid SCHEMBL588103 0.78 LMNA (0.79) KCNH2HRH1OPRK1ADORA3CNR1
Hydrochloric Acid SCHEMBL588128 0.78 LMNA (0.79) KCNH2HRH1OPRK1ADORA3CNR1
Hydrochloric Acid SCHEMBL587709 0.78 LMNA (0.79) KCNH2HRH1OPRK1ADORA3CNR1
SCHEMBL8556503 0.78 SIGMAR1 (0.58) KCNH2LMNADRD3DRD2CYP3A4
SCHEMBL7668121 0.76 CHRM2 (0.83) KCNH2HRH1OPRK1ADORA3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883622-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1998-12-16 EP claimed
WO-1997031923-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1997-09-04 WO claimed
EP-0883622-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1998-12-16 EP disclosed
WO-1997031923-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1997-09-04 WO disclosed