SCHEMBL8556735

SCHEMBL8556735

Cc1c(CCC(=O)O)nc2c(=O)[nH]c3ccc(Cl)cc3n12

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.48
EGFR P00533 1/20 0.43
FFAR1 O14842 2/20 0.41
PPARG P37231 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ADORA1 P30542 1/20 0.40
GPR17 Q13304 1/20 0.40
KMO O15229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558994 0.88 ADORA3 (0.55) ADORA3EGFRKDM4EALDH1A1ADORA1
SCHEMBL8558992 0.83 CHEK1 (0.44) ADORA3KDM4EALDH1A1
SCHEMBL8553602 0.81 PDE5A (0.41) ALDH1A1KMO
SCHEMBL8559477 0.80 CHEK1 (0.51)
SCHEMBL8554829 0.78 PDE9A (0.61) PPARGGPR17KMO
SCHEMBL8557272 0.77 CHEK1 (0.44) ADORA3KDM4E
SCHEMBL3599601 0.76 ADORA3 (0.43) ADORA3FFAR1PPARGGPR17KMO
SCHEMBL8558719 0.76 ADORA3 (0.50) ADORA3EGFRADORA1
SCHEMBL3600026 0.75 PDE9A (0.43) ADORA3FFAR1PPARGKDM4EALDH1A1
SCHEMBL8556228 0.74 ADORA3 (0.50) ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691970-B1 IMIDAZOLOQUINOXALINONE DERIVATIVES AS EAA ANTAGONISTS BASF AG (DE) 1998-11-11 EP disclosed